KEGG   DGROUP: ABCB1 substrate
Entry
DG01665                     DGroup                                 
Name
ABCB1 substrate
Type
Metabolism
Member
Odevixibat
 D11716  
Odevixibat (USAN)
 D13092  
Odevixibat hydrate (JAN)  <US>
D02554  
Rifaximin (JAN/USAN/INN)  <JP/US>
Loperamide
 D08144  
Loperamide (INN)
 D00729  
Loperamide hydrochloride (JAN/USP)  <JP/US>
 D07113  
Loperamide oxide (INN)
D10264  
Linagliptin and metformin hydrochloride  <US>
D10588  
Empagliflozin and linagliptin  <JP/US>
D09592  
Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN)  <JP/US>
D10459  
Empagliflozin (JAN/USAN/INN)  <JP/US>
Eliglustat
 D09893  
Eliglustat (USAN/INN)
 D09894  
Eliglustat tartrate (JAN/USAN)  <JP/US>
D04768  
Lonafarnib (JAN/USAN/INN)  <JP/US>
D09017  
Ticagrelor (JAN/USAN/INN)  <JP/US>
Dabigatran
 D09707  
Dabigatran (USAN/INN)
 D07144  
Dabigatran etexilate (USAN/INN)
 D07082  
Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN)  <JP/US>
D07086  
Rivaroxaban (JAN/USAN/INN)  <JP/US>
D03213  
Apixaban (JAN/USAN/INN)  <JP/US>
Edoxaban
 D09710  
Edoxaban (USAN/INN)
 D09546  
Edoxaban tosilate hydrate (JAN)  <JP/US>
 D11568  
Edoxaban tosylate (USAN)
Berotralstat
 D11673  
Berotralstat (USAN/INN)
 D11674  
Berotralstat hydrochloride (JAN/USAN)  <JP/US>
D00297  
Digitoxin (JAN/USP/INN)
D00298  
Digoxin (JP18/USP)  <JP/US>
Metildigoxin
 D09847  
Metildigoxin (INN); Medigoxin (BAN)
 D02587  
Metildigoxin (JP18)  <JP>
Ranolazine
 D05700  
Ranolazine (USAN/INN)  <US>
 D05701  
Ranolazine hydrochloride (USAN)
D09572  
Riociguat (JAN/USAN/INN)  <JP/US>
D01213  
Tolvaptan (JP18/USAN/INN)  <JP/US>
Verapamil
 D02356  
Verapamil (USAN/INN)
 D00619  
Verapamil hydrochloride (JP18/USP)  <JP/US>
Olmesartan
 D05246  
Olmesartan (USAN/INN)
 D01204  
Olmesartan medoxomil (JP18/USP)  <JP/US>
Aliskiren
 D03208  
Aliskiren (USAN/INN)
 D06412  
Aliskiren fumarate (JAN/USAN)  <JP/US>
Atorvastatin
 D07474  
Atorvastatin (INN)  <US>
 D00887  
Atorvastatin calcium anhydorous
 D02258  
Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18)  <JP/US>
 D11095  
Atorvastatin calcium propylene glycol solvate  <US>
D01966  
Ezetimibe (JAN/USP/INN)  <JP/US>
D00804  
Ivermectin (JAN/USP/INN)  <JP/US>
D10433  
Vibegron (JAN/USAN/INN)  <JP/US>
D03671  
Deflazacort (USAN/INN)  <US>
Azithromycin
 D07486  
Azithromycin (INN)  <US>
 D02134  
Azithromycin hydrate (JP18)  <JP/US>
 D06390  
Azithromycin (USP)  <US>
D02555  
Posaconazole (JAN/USAN/INN)  <JP/US>
Saquinavir
 D00429  
Saquinavir (JAN/USP/INN)
 D01160  
Saquinavir mesylate (USP); Saquinavir mesilate (JAN)
D10428  
Tenofovir alafenamide (USAN/INN)
D10605  
Tenofovir alafenamide fumarate (JAN/USAN)  <JP/US>
Simeprevir
 D10081  
Simeprevir (JAN/USAN)
 D10469  
Simeprevir sodium (JAN)
D10093  
Asunaprevir (JAN/USAN)
Daclatasvir
 D10065  
Daclatasvir (USAN)
 D10105  
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN)
D10366  
Sofosbuvir (JAN/USAN/INN)  <US>
D10625  
Elbasvir (JAN/USAN/INN)
Grazoprevir
 D11565  
Grazoprevir (USAN/INN)
 D10639  
Grazoprevir (USAN); Grazoprevir hydrate (JAN)
D10578  
Ledipasvir and sofosbuvir  <JP/US>
D10582  
Dasabuvir, ombitasvir, paritaprevir and ritonavir
D10745  
Ombitasvir, paritaprevir and ritonavir
D10827  
Sofosbuvir and velpatasvir  <JP/US>
D11014  
Glecaprevir and pibrentasvir  <JP/US>
D10882  
Daclatasvir, asunaprevir and beclabuvir
D10835  
Emtricitabine and tenofovir alafenamide  <JP/US>
D10755  
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide  <JP/US>
D10836  
Emtricitabine, rilpivirine and tenofovir alafenamide  <JP/US>
D11382  
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide  <JP/US>
Lenacapavir
 D12161  
Lenacapavir (USAN/INN)
 D12162  
Lenacapavir sodium (JAN/USAN)  <JP/US>
Topotecan
 D08618  
Topotecan (BAN)
 D02168  
Topotecan hydrochloride (USAN); Nogitecan hydrochloride (JAN)  <JP/US>
Nilotinib
 D08953  
Nilotinib (USAN/INN)
 D06413  
Nilotinib hydrochloride hydrate (JAN)  <JP/US>
 D12444  
Nilotinib hydrochloride dihydrate (JAN)
 D12854  
Nilotinib laurylsulfate (USAN)
 D13008  
Nilotinib D-tartrate (USAN)  <US>
Afatinib
 D09724  
Afatinib (USAN/INN)
 D09733  
Afatinib dimaleate (USAN); Afatinib maleate (JAN)  <JP/US>
D02714  
Everolimus (JAN/USAN/INN)  <JP/US>
D00753  
Sirolimus (JAN/USAN/INN)  <JP/US>
Lapatinib
 D08108  
Lapatinib (INN)
 D04024  
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN)  <JP/US>
D10927  
Erdafitinib (JAN/USAN/INN)  <JP/US>
Regorafenib
 D10138  
Regorafenib (USAN/INN)
 D10137  
Regorafenib hydrate (JAN)  <JP/US>
Lenvatinib
 D09919  
Lenvatinib (USAN/INN)
 D09920  
Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN)  <JP/US>
Nintedanib
 D10481  
Nintedanib (USAN/INN)
 D10396  
Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN)  <JP/US>
Gilteritinib
 D10709  
Gilteritinib (USAN/INN)
 D10800  
Gilteritinib fumarate (JAN/USAN)  <JP/US>
Tazemetostat
 D11444  
Tazemetostat (USAN/INN)
 D11485  
Tazemetostat hydrobromide (JAN/USAN)  <JP/US>
D10888  
Relugolix (JAN/USAN/INN)  <JP/US>
D10308  
Baricitinib (JAN/USAN/INN)  <JP/US>
D00570  
Colchicine (JP18/USP)  <JP/US>
D10915  
Cannabidiol (JAN/USAN/INN)  <US>
Citalopram
 D07704  
Citalopram (USP/INN)
 D00822  
Citalopram hydrobromide (USP)  <US>
 D07705  
Citalopram hydrochloride
Methadone
 D08195  
Methadone (BAN)
 D02102  
Methadone hydrochloride (JAN/USP)  <JP/US>
Quinine
 D08460  
Quinine (BAN)
 D01663  
Quinine ethylcarbonate (JP18)
 D02261  
Quinine hydrochloride hydrate (JP18)
 D02262  
Quinine sulfate (USP); Quinine sulfate hydrate (JP18)  <US>
 D05681  
Quinine ascorbate (USAN)
 D08461  
Quinine dihydrochloride
Indacaterol
 D09318  
Indacaterol (USAN/INN)
 D09319  
Indacaterol maleate (JAN/USAN)  <JP>
 D11009  
Indacaterol acetate (JAN)
D10505  
Glycopyrronium bromide and indacaterol maleate  <JP>
Cetirizine
 D07662  
Cetirizine (INN)
 D00664  
Cetirizine hydrochloride (JP18/USP)  <JP/US>
D10897  
Teneligliptin and canagliflozin  <JP>
Temsavir
 D10734  
Temsavir (USAN/INN)
 D10707  
Fostemsavir (USAN)
 D10708  
Fostemsavir tromethamine (USAN)  <US>
 » expand
Class
Transporter substrate
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